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Literature summary for 3.4.22.52 extracted from

  • Passiatore, G.; Rom, S.; Eletto, D.; Peruzzi, F.
    HIV-1 Tat C-terminus is cleaved by calpain 1: implication for Tat-mediated neurotoxicity (2009), Biochim. Biophys. Acta, 1793, 378-387.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
acetyl-calpastatin peptide 50 microM Rattus norvegicus
lactacystin 1 microM Rattus norvegicus
MG115 inhibitory effect in micromolar concentrations, 1 mircoM Rattus norvegicus
MG132 inhibitory effect in micromolar concentrations, 1 microM Rattus norvegicus
N-acetyl-Leu-Leu-norleucinal 2-fold increase in Tat levels after pre-treating with ALLN, 10 microM Rattus norvegicus

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+
-
Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Rattus norvegicus

Source Tissue

Source Tissue Comment Organism Textmining
neuronal cell line progenitor HCN-A94-2 Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
RecTat101 + H2O
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
calpain 1
-
Rattus norvegicus