Application | Comment | Organism |
---|---|---|
medicine | enzyme has potential as a sensitive and early tumor marker | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
iodoacetamide | - |
Homo sapiens | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | ie.e. E-64 | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.027 | - |
D-Ile-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.061 | - |
N-p-tosyl-Gly-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.109 | - |
D-Ala-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.153 | - |
N-p-tosyl-Gly-Pro-Lys-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.306 | - |
Glu-Glu-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
factor X + H2O | Homo sapiens | cleavage of Arg-Ile bond, activation of the coaglutation factor X | factor Xa | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
to homogeneity | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
amnion | - |
Homo sapiens | - |
chorion | - |
Homo sapiens | - |
additional information | produced by malignant and fetal cells | Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Homo sapiens |
47 | - |
purified enzyme | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
benzyloxycarbonyl-Arg-Arg-4-nitroanilide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Arg-Arg + 4-nitroaniline | - |
? | |
benzyloxycarbonyl-Leu-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Leu-Pro-Arg + 4-nitroaniline | - |
? | |
benzyloxycarbonyl-Val-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Val-Pro-Arg + 4-nitroaniline | - |
? | |
D-Ala-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | D-Ala-Pro-Arg + 4-nitroaniline | - |
? | |
D-Ile-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | D-Ile-Pro-Arg + 4-nitroaniline | - |
? | |
D-Phe-Pip-Arg-4-nitroanilide + H2O | - |
Homo sapiens | D-Phe-Pip-Arg + 4-nitroaniline | - |
? | |
factor X + H2O | cleavage of Arg-Ile bond | Homo sapiens | factor Xa | - |
? | |
factor X + H2O | cleavage of Arg-Ile bond, activation of the coaglutation factor X | Homo sapiens | factor Xa | - |
? | |
Fibrinogen + H2O | - |
Homo sapiens | ? | - |
? | |
Glu-Glu-Phe-Lys-4-nitroanilide + H2O | - |
Homo sapiens | Glu-Glu-Phe-Lys + 4-nitroaniline | - |
? | |
Glu-Glu-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | Glu-Glu-Pro-Arg + 4-nitroaniline | - |
? | |
Leu-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | Leu-Pro-Arg + 4-nitroaniline | - |
? | |
methylsulfonyl-D-cyclohexylalanyl-butyl-Arg-4-nitroanilide + H2O | - |
Homo sapiens | methylsulfonyl-D-cyclohexylalanyl-butyl-Arg + 4-nitroaniline | - |
? | |
additional information | substrate specificity, overview | Homo sapiens | ? | - |
? | |
N-p-tosyl-Gly-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | N-p-tosyl-Gly-Pro-Arg + 4-nitroaniline | - |
? | |
N-p-tosyl-Gly-Pro-Lys-4-nitroanilide + H2O | - |
Homo sapiens | N-p-tosyl-Gly-Pro-Lys + 4-nitroaniline | - |
? | |
sarcosyl-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | sarcosyl-Pro-Arg + 4-nitroaniline | - |
? | |
Val-Pro-Arg-4-nitroanilide + H2O | - |
Homo sapiens | Val-Pro-Arg + 4-nitroaniline | - |
? |
Synonyms | Comment | Organism |
---|---|---|
cancer procoagulant | - |
Homo sapiens |
CP | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0073 | - |
N-p-tosyl-Gly-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.0082 | - |
D-Ile-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.0119 | - |
Glu-Glu-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.0129 | - |
N-p-tosyl-Gly-Pro-Lys-4-nitroanilide | pH 7.2 | Homo sapiens | |
0.0132 | - |
D-Ala-Pro-Arg-4-nitroanilide | pH 7.2 | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.2 | - |
assay at | Homo sapiens |