Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Benzyloxycarbonyl-Phe-Phe-CHN2 | - |
Bos taurus | |
Benzyloxycarbonyl-Phe-Phe-CHN2 | - |
Homo sapiens | |
Benzyloxycarbonyl-Phe-Phe-CHN2 | - |
Oryctolagus cuniculus | |
Benzyloxycarbonyl-Phe-Phe-CHN2 | - |
Ovis aries | |
Benzyloxycarbonyl-Phe-Phe-CHN2 | - |
Rattus norvegicus | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Bos taurus | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Homo sapiens | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Oryctolagus cuniculus | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Ovis aries | |
trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0018 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Oryctolagus cuniculus | |
0.0018 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Ovis aries | |
0.0022 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Bos taurus | |
0.0024 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Homo sapiens | |
0.0045 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
ox | - |
Homo sapiens | - |
- |
- |
Oryctolagus cuniculus | - |
- |
- |
Ovis aries | - |
- |
- |
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | ? | - |
? | |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Rattus norvegicus | ? | - |
? | |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Bos taurus | ? | - |
? | |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Oryctolagus cuniculus | ? | - |
? | |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Ovis aries | ? | - |
? |
Subunits | Comment | Organism |
---|---|---|
dimer | 1 * 22000-25000 + 1 * 5000-7000, SDS-PAGE under reducing conditions | Homo sapiens |
dimer | 1 * 22000-25000 + 1 * 5000-7000, SDS-PAGE under reducing conditions | Rattus norvegicus |
dimer | 1 * 22000-25000 + 1 * 5000-7000, SDS-PAGE under reducing conditions | Bos taurus |
dimer | 1 * 22000-25000 + 1 * 5000-7000, SDS-PAGE under reducing conditions | Oryctolagus cuniculus |
dimer | 1 * 22000-25000 + 1 * 5000-7000, SDS-PAGE under reducing conditions | Ovis aries |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
10 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Homo sapiens | |
17 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Homo sapiens | |
20 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Oryctolagus cuniculus | |
26 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Rattus norvegicus | |
30 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Ovis aries |