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Literature summary for 3.4.21.75 extracted from

  • Angliker, H.; Neumann, U.; Molloy, S.S.; Thomas, G.
    Internally quenched fluorogenic substrate for furin (1995), Anal. Biochem., 224, 409-412.
    View publication on PubMed

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.002
-
protective antigen (-Arg-Lys-Lys-Arg-Ser-Thr-Ser-Ala-Gly-) Mammalia
0.0038
-
2-Aminobenzoyl-Arg-Val-Lys-Arg-Gly-Leu-Ala-Tyr(NO2)-Asp-OH
-
Mammalia
0.0156
-
tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide
-
Mammalia

Organism

Organism UniProt Comment Textmining
Mammalia
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2-Aminobenzoyl-Arg-Val-Lys-Arg-Gly-Leu-Ala-Tyr(NO2)-Asp-OH + H2O
-
Mammalia ?
-
?
protective antigen + H2O
-
Mammalia ?
-
?
tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide + H2O
-
Mammalia tert-butoxycarbonyl-Arg-Val-Arg-Arg + 7-amino-4-methylcoumarin
-
?

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Mammalia

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
0.192
-
tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide
-
Mammalia
11
-
protective antigen (-Arg-Lys-Lys-Arg-Ser-Thr-Ser-Ala-Gly-) Mammalia
29.3
-
2-Aminobenzoyl-Arg-Val-Lys-Arg-Gly-Leu-Ala-Tyr(NO2)-Asp-OH
-
Mammalia