Inhibitors | Comment | Organism | Structure |
---|---|---|---|
concanavalin A | - |
Homo sapiens | |
plasminogen activator inhibitor 1 | phosphorylated uPA is less sensitive to inhibition than nonphosphorylated uPA | Homo sapiens | |
Plasminogen activator inhibitor 2 | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000243 | - |
plasminogen | pH 7.5, nonphosphorylated uPA | Homo sapiens | |
0.017 | - |
plasminogen | pH 7.5, phosphorylated uPA | Homo sapiens | |
0.297 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 8.8, phosphorylated uPA | Homo sapiens | |
0.392 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 7.5, phosphorylated uPA | Homo sapiens | |
0.438 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 8.8, nonphosphorylated uPA | Homo sapiens | |
0.608 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 7.5, nonphosphorylated uPA | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
A-431 cell | - |
Homo sapiens | - |
Detroit 562 cell | - |
Homo sapiens | - |
ECV304 cell | - |
Homo sapiens | - |
urine | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-diglutamyl-glycyl-L-arginine-4-nitroanilide + H2O | - |
Homo sapiens | L-diglutamyl-glycyl-L-arginine + 4-nitroaniline | - |
? | |
plasminogen + H2O | - |
Homo sapiens | plasmin + ? | generation of 2 polypeptides, one of 80000 MW (A-chain), and the other of 27000 MW (B-chain) | ? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0075 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 8.8, nonphosphorylated uPA | Homo sapiens | |
0.0113 | - |
L-diglutamyl-glycyl-L-arginine-4-nitroanilide | pH 7.5, nonphosphorylated uPA | Homo sapiens | |
0.0383 | - |
plasminogen | pH 7.5, nonphosphorylated uPA | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | 9.5 | phosphorylated uPA | Homo sapiens |
8.8 | 9.5 | nonphosphorylated uPA | Homo sapiens |