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Literature summary for 3.4.21.37 extracted from

  • Ying, Q.L.; Simon, S.R.
    Kinetics of the inhibition of human leukocyte elastase by elafin, a 6-kilodalton elastase-specific inhibitor from human skin (1993), Biochemistry, 32, 1866-1874.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
elafin a potent, substratelike, but fully reversible inhibitor Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
azurophil granule
-
Homo sapiens 42582
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
neutrophil
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Nalpha-methoxysuccinyl-Nepsilon-2-picolinoyl-L-lysinyl-L-Ala-L-Pro-L-Val 4-nitroanilide + H2O
-
Homo sapiens ?
-
?

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000017
-
elafin pH 8.0, 25°C Homo sapiens
0.0000002
-
elafin pH 9.0, 25°C Homo sapiens
0.0000067
-
elafin pH 5.4, 25°C Homo sapiens