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Literature summary for 3.4.21.36 extracted from

  • Kwan, J.C.; Taori, K.; Paul, V.J.; Luesch, H.
    Lyngbyastatins 8-10, elastase inhibitors with cyclic depsipeptide scaffolds isolated from the marine cyanobacterium Lyngbya semiplena (2009), Mar. Drugs, 7, 528-538.
    View publication on PubMedView publication on EuropePMC
Search for more literature for 3.4.21.36

Inhibitors

Inhibitors Comment Organism Structure
lyngbyastatin 10
-
 Sus scrofa
lyngbyastatin 7
-
 Sus scrofa
lyngbyastatin 8
-
 Sus scrofa
lyngbyastatin 9
-
 Sus scrofa

Organism

Organism UniProt Comment Textmining
Sus scrofa
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
pancreas
-
 Sus scrofa
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
succinyl-L-Ala-L-Ala-L-Ala-4-nitroanilide + H2O
-
 Sus scrofa ?
-
 ?

Synonyms

Synonyms Comment Organism
elastase
-
 Sus scrofa

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0000473
-
 in Tris-HCl (pH 8.0) Sus scrofa lyngbyastatin 7
0.00012
-
 in Tris-HCl (pH 8.0) Sus scrofa lyngbyastatin 10
0.000123
-
 in Tris-HCl (pH 8.0) Sus scrofa lyngbyastatin 8
0.00021
-
 in Tris-HCl (pH 8.0) Sus scrofa lyngbyastatin 9