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Literature summary for 3.4.21.109 extracted from

  • List, K.
    Matriptase: a culprit in cancer? (2009), Future Oncol., 5, 97-104.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information autoactivation Mus musculus
additional information autoactivation Homo sapiens

Application

Application Comment Organism
medicine matriptase is identified as a cancer-associated protease Mus musculus
medicine matriptase is identified as a cancer-associated protease Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
alpha-1-antitrypsin
-
Homo sapiens
alpha-1-antitrypsin
-
Mus musculus
alpha-2-Antiplasmin
-
Homo sapiens
alpha-2-Antiplasmin
-
Mus musculus
antithrombin III
-
Homo sapiens
antithrombin III
-
Mus musculus
hepatocyte growth factor activator inhibitor-1 HAI-1 Homo sapiens
hepatocyte growth factor activator inhibitor-1 HAI-1 Mus musculus
hepatocyte growth factor activator inhibitor-2 HAI-2 Homo sapiens
hepatocyte growth factor activator inhibitor-2 HAI-2 Mus musculus

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane
-
Mus musculus 16020
-
membrane
-
Homo sapiens 16020
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
CDCP1 + H2O Mus musculus
-
?
-
?
CDCP1 + H2O Homo sapiens
-
?
-
?
G-protein-coupled protease-activated receptor-2 + H2O Mus musculus
-
?
-
?
G-protein-coupled protease-activated receptor-2 + H2O Homo sapiens
-
?
-
?
growth factor macrophage-stimulating protein 1 + H2O Mus musculus
-
?
-
?
growth factor macrophage-stimulating protein 1 + H2O Homo sapiens
-
?
-
?
insulin-like growth factor binding-related protein-1 + H2O Mus musculus
-
?
-
?
insulin-like growth factor binding-related protein-1 + H2O Homo sapiens
-
?
-
?
pro-hepatocyte growth factor + H2O Mus musculus
-
?
-
?
pro-hepatocyte growth factor + H2O Homo sapiens
-
?
-
?
pro-urokinase-type plasminogen activator + H2O Mus musculus
-
?
-
?
pro-urokinase-type plasminogen activator + H2O Homo sapiens
-
?
-
?
prostatin + H2O Mus musculus
-
?
-
?
prostatin + H2O Homo sapiens
-
?
-
?
SIMA135 + H2O Mus musculus
-
?
-
?
SIMA135 + H2O Homo sapiens
-
?
-
?
trask + H2O Mus musculus
-
?
-
?
trask + H2O Homo sapiens
-
?
-
?
VEGFR-2 + H2O Mus musculus
-
?
-
?
VEGFR-2 + H2O Homo sapiens
-
?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
epithelial cell
-
Mus musculus
-
epithelial cell
-
Homo sapiens
-
macrophage
-
Mus musculus
-
macrophage
-
Homo sapiens
-
mast cell
-
Mus musculus
-
mast cell
-
Homo sapiens
-
monocyte
-
Mus musculus
-
monocyte
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
CDCP1 + H2O
-
Mus musculus ?
-
?
CDCP1 + H2O
-
Homo sapiens ?
-
?
G-protein-coupled protease-activated receptor-2 + H2O
-
Mus musculus ?
-
?
G-protein-coupled protease-activated receptor-2 + H2O
-
Homo sapiens ?
-
?
growth factor macrophage-stimulating protein 1 + H2O
-
Mus musculus ?
-
?
growth factor macrophage-stimulating protein 1 + H2O
-
Homo sapiens ?
-
?
insulin-like growth factor binding-related protein-1 + H2O
-
Mus musculus ?
-
?
insulin-like growth factor binding-related protein-1 + H2O
-
Homo sapiens ?
-
?
pro-hepatocyte growth factor + H2O
-
Mus musculus ?
-
?
pro-hepatocyte growth factor + H2O
-
Homo sapiens ?
-
?
pro-urokinase-type plasminogen activator + H2O
-
Mus musculus ?
-
?
pro-urokinase-type plasminogen activator + H2O
-
Homo sapiens ?
-
?
prostatin + H2O
-
Mus musculus ?
-
?
prostatin + H2O
-
Homo sapiens ?
-
?
SIMA135 + H2O
-
Mus musculus ?
-
?
SIMA135 + H2O
-
Homo sapiens ?
-
?
trask + H2O
-
Mus musculus ?
-
?
trask + H2O
-
Homo sapiens ?
-
?
VEGFR-2 + H2O
-
Mus musculus ?
-
?
VEGFR-2 + H2O
-
Homo sapiens ?
-
?

Synonyms

Synonyms Comment Organism
epithin
-
Mus musculus
epithin
-
Homo sapiens
matriptase
-
Mus musculus
matriptase
-
Homo sapiens
MT-SP1
-
Mus musculus
MT-SP1
-
Homo sapiens
ST14
-
Mus musculus
ST14
-
Homo sapiens
TADG-15
-
Mus musculus
TADG-15
-
Homo sapiens
type II transmembrane serine protease
-
Mus musculus
type II transmembrane serine protease
-
Homo sapiens