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Literature summary for 3.4.21.109 extracted from

  • Jiang, S.; Li, P.; Lee, S.L.; Lin, C.Y.; Long, Y.Q.; Johnson, M.D.; Dickson, R.B.; Roller, P.P.
    Design and synthesis of redox stable analogues of sunflower trypsin inhibitors (SFTI-1) on solid support, potent inhibitors of matriptase (2007), Org. Lett., 9, 9-12.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
additional information inhibitor synthesis and validation, overview Homo sapiens
sunflower trypsin inhibitor-1 SFTI-1, isolated from sunflower seeds Homo sapiens
sunflower trypsin inhibitor-2 SFTI-2 Homo sapiens
sunflower trypsin inhibitor-3 SFTI-3 Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane matriptase is a type II transmembrane protein Homo sapiens 16020
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Synonyms

Synonyms Comment Organism
More matriptase is a member of the type II transmembrane serine protease family Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000092
-
sunflower trypsin inhibitor-1
-
Homo sapiens
0.0000025
-
sunflower trypsin inhibitor-3
-
Homo sapiens
0.000025
-
sunflower trypsin inhibitor-2
-
Homo sapiens