Application | Comment | Organism |
---|---|---|
analysis | mass spectrometric assay for angiotensin-converting enzyme 2 using angiotensin II as substrate will have applications in drug screening, antagonist development, and clinical investigations | Mus musculus |
analysis | mass spectrometric assay for angiotensin-converting enzyme 2 using angiotensin II as substrate will have applications in drug screening, antagonist development, and clinical investigations | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
MLN 4760 | IC50: 3 nM | Homo sapiens | |
MLN 4760 | IC50: 3 nM | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
recombinant | - |
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Mus musculus | - |
additional information | no activity in plasma | Mus musculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
angiotensin II + H2O | - |
Mus musculus | angiotensin-(1-7) + Phe | - |
? | |
angiotensin II + H2O | - |
Homo sapiens | angiotensin-(1-7) + Phe | - |
? | |
additional information | angiotensin I is not a good substrate for recombinant human ACE2 | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ACE2 | - |
Mus musculus |
ACE2 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000003 | - |
IC50: 3 nM | Mus musculus | MLN 4760 | |
0.000003 | - |
IC50: 3 nM | Homo sapiens | MLN 4760 |