Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | 1 mM, 90% inhibition | Rattus norvegicus | |
2-oxoglutarate | 0.1 mM, 46% inhibition | Rattus norvegicus | |
Ala-Glu | 0.0061 mM, 50% inhibition | Rattus norvegicus | |
Asp-Ala | 0.1 mM, 26% inhibition | Rattus norvegicus | |
Asp-Asp | 0.1 mM, 42% inhibition | Rattus norvegicus | |
Asp-Glu | 0.0024 mM, 50% inhibition | Rattus norvegicus | |
Asp-Phe | 0.1 mM, 22% inhibition | Rattus norvegicus | |
aspartate | 0.1 mM, 42% inhibition | Rattus norvegicus | |
bestatin | 0.29 mM, 79% inhibition | Rattus norvegicus | |
Cd2+ | - |
Rattus norvegicus | |
Cu2+ | - |
Rattus norvegicus | |
cysteate | 0.1 mM, 40% inhibition | Rattus norvegicus | |
cysteine sulfinate | 0.1 mM, 42% inhibition | Rattus norvegicus | |
D-Glu-D-Glu | 0.1 mM, 50% inhibition | Rattus norvegicus | |
dithiothreitol | 1 mM, 94.8% inhibition | Rattus norvegicus | |
EDTA | 1 mM, 96.3% inhibition | Rattus norvegicus | |
EGTA | 1 mM, 92% inhibition | Rattus norvegicus | |
Fe3+ | - |
Rattus norvegicus | |
gamma-Glu-Glu | 0.0095 mM, 50% inhibition | Rattus norvegicus | |
Glu-Asp | 0.1 mM, 27% inhibition | Rattus norvegicus | |
Glu-Glu | 0.00075 mM, 50% inhibition | Rattus norvegicus | |
Glu-Glu-Glu | 0.062 mM, 50% inhibition | Rattus norvegicus | |
glutathione | i.e. gamma-Glu-Cys-Gly, 0.019 mM, 50% inhibition | Rattus norvegicus | |
Gly-Glu | 0.008 mM, 50% inhibition | Rattus norvegicus | |
Gly-Gly-Glu | 0.00098 mM, 50% inhibition | Rattus norvegicus | |
Ibotenate | 0.1 mM, 45% inhibition | Rattus norvegicus | |
iodoacetate | 1 mM, 38% inhibition | Rattus norvegicus | |
L-2-Amino-4-phosphonobutanoate | 0.1 mM, 37% inhibition | Rattus norvegicus | |
L-Glu | 0.032 mM, 50% inhibition | Rattus norvegicus | |
additional information | not inhibitory are pepstatin, iodoacetamide, amastatin | Rattus norvegicus | |
N-Acetyl-Asp-Gln | 0.1 mM, 49% inhibition | Rattus norvegicus | |
N-Acetyl-Asp-Glu-Asp | 0.1 mM, 49% inhibition | Rattus norvegicus | |
N-Acetyl-Asp-Ser-Gly | 0.1 mM, 37% inhibition | Rattus norvegicus | |
N-Acetyl-Glu-Asp | 0.036 mM, 50% inhibition | Rattus norvegicus | |
N-Acetyl-Glu-Glu | 0.00031 mM, 50% inhibition | Rattus norvegicus | |
N-acetyl-L-Asp | 0.1 mM, 38% inhibition | Rattus norvegicus | |
N-Acetyl-L-Asp-L-Glu | 0.00054 mM, 50% inhibition | Rattus norvegicus | |
N-acetyl-L-Glu | 0.058 mM, 50% inhibition | Rattus norvegicus | |
Phe-Glu | 0.077 mM, 50% inhibition | Rattus norvegicus | |
PO43- | - |
Rattus norvegicus | |
puromycin | 0.5 mM, 55% inhibition | Rattus norvegicus | |
pyroglutamate | 0.1 mM, 27% inhibition | Rattus norvegicus | |
quinolinate | 0.1 mM, 41% inhibition | Rattus norvegicus | |
Quisqualic acid | 0.00048 mM, 50% inhibition | Rattus norvegicus | |
Serine O-sulfate | 0.042 mM, 50% inhibition | Rattus norvegicus | |
SO42- | - |
Rattus norvegicus | |
Tyr-Glu | 0.1 mM, 45% inhibition | Rattus norvegicus | |
Val-Glu-Glu | 0.036 mM, 50% inhibition | Rattus norvegicus | |
Zn2+ | - |
Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
540 | - |
N-Acetyl-L-Asp-L-Glu | - |
Rattus norvegicus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Rattus norvegicus | 16020 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Br- | 2 mM, activation | Rattus norvegicus | |
Ca2+ | activation | Rattus norvegicus | |
Cl- | 2 mM, activation | Rattus norvegicus | |
Co2+ | activation | Rattus norvegicus | |
F- | 100 mM, 20% of the activity compared to Cl- | Rattus norvegicus | |
I- | 2 mM, activation | Rattus norvegicus | |
Mg2+ | activation | Rattus norvegicus | |
Mn2+ | activation | Rattus norvegicus | |
NO3- | 2 mM , activation | Rattus norvegicus | |
Sr2+ | activation | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | forebrain | Rattus norvegicus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
assay method | Rattus norvegicus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N-Acetyl-L-Asp-L-Glu + H2O | - |
Rattus norvegicus | N-Acetyl-L-Asp + L-Glu | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
- |
Rattus norvegicus |
Temperature Minimum [°C] | Temperature Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | 80 | more than 50% of maximal activity in this range | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7 | - |
- |
Rattus norvegicus |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
6 | 7.4 | more than 50% of maximal activity in this range | Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00031 | - |
N-Acetyl-Glu-Glu | - |
Rattus norvegicus | |
0.00054 | - |
N-Acetyl-L-Asp-L-Glu | - |
Rattus norvegicus | |
0.00075 | - |
Glu-Glu | - |
Rattus norvegicus | |
0.00098 | - |
Gly-Gly-Glu | - |
Rattus norvegicus | |
0.0024 | - |
Asp-Glu | - |
Rattus norvegicus | |
0.008 | - |
Gly-Glu | - |
Rattus norvegicus | |
0.019 | - |
glutathione | i.e. gamma-Glu-Cys-Gly | Rattus norvegicus | |
0.036 | - |
N-Acetyl-Glu-Asp | - |
Rattus norvegicus | |
0.036 | - |
Val-Glu-Glu | - |
Rattus norvegicus | |
0.042 | - |
Serine O-sulfate | - |
Rattus norvegicus | |
0.058 | - |
N-acetyl-L-Glu | - |
Rattus norvegicus | |
0.061 | - |
Ala-Glu | - |
Rattus norvegicus | |
0.062 | - |
Glu-Glu-Glu | - |
Rattus norvegicus | |
0.077 | - |
Phe-Glu | - |
Rattus norvegicus | |
0.095 | - |
gamma-Glu-Glu | - |
Rattus norvegicus | |
0.1 | - |
D-Glu-D-Glu | - |
Rattus norvegicus |