Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | - |
Bos taurus | |
2-D-Methylsuccinyl-L-Pro | - |
Bos taurus | |
3-Mercaptopropanoyl-L-Pro | - |
Bos taurus | |
bradykinin potentiating factor | - |
Bos taurus | |
D-2-Methyl-3-mercaptopropanoyl-L-Pro | i.e. captopril | Bos taurus | |
DTT | - |
Bos taurus | |
EDTA | - |
Bos taurus | |
mercaptoethanol | - |
Bos taurus | |
additional information | marked substrate inhibition with benzoyl-Gly-His-Leu, but little or no substrate inhibition with benzoyl-Gly-His-Gly; the enzyme is 5500 times less sensitive to D-Cys-L-Pro, the very potent inhibitor of angiotensin I-converting enzyme (EC 3.4.15.1) | Bos taurus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.8 | - |
benzoyl-Gly-His-Leu | - |
Bos taurus | |
2.4 | - |
benzoyl-Gly-His-Gly | - |
Bos taurus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Bos taurus | 16020 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
additional information | in contrast to peptidyl-dipeptidase A (EC 3.4.15.1) it displays no dependence on Cl- | Bos taurus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
240000 | - |
bovine, sucrose density gradient sedimentation, gel filtration | Bos taurus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
partial | Bos taurus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
atrium | - |
Bos taurus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Bos taurus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Atriopeptin II + H2O | - |
Bos taurus | Atriopeptin I + ? | - |
? | |
benzoyl-Gly-His-Gly + H2O | - |
Bos taurus | benzoyl-Gly + His-Gly | - |
? | |
benzoyl-Gly-His-Leu + H2O | - |
Bos taurus | ? | - |
? |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.3 | - |
- |
Bos taurus |