Inhibitors | Comment | Organism | Structure |
---|---|---|---|
bestatin | non-competitive | Homo sapiens | |
Cilastatin | competitive | Homo sapiens | |
DTT | reversible, competitive | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.09 | - |
L-Val-Gly | - |
Homo sapiens | |
0.15 | - |
L-Trp-Gly | - |
Homo sapiens | |
0.21 | - |
L-Leu-Gly | - |
Homo sapiens | |
0.67 | - |
L-Phe-Gly | - |
Homo sapiens | |
0.99 | - |
Gly-L-Phe | - |
Homo sapiens | |
1.22 | - |
Gly-L-Leu | - |
Homo sapiens | |
2.03 | - |
Gly-L-Trp | - |
Homo sapiens | |
11 | - |
Gly-L-Val | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Gly-Leu + H2O | - |
Homo sapiens | Gly + Leu | - |
? | |
Gly-Phe + H2O | - |
Homo sapiens | Gly + Phe | - |
? | |
Gly-Trp + H2O | - |
Homo sapiens | Gly + Trp | - |
? | |
Gly-Val + H2O | - |
Homo sapiens | Gly + Val | - |
? | |
Leu-Gly + H2O | - |
Homo sapiens | Leu + Gly | - |
? | |
additional information | enzyme prefers substrates with bulky, hydrophobic group of the dipeptide located at the N-terminal position | Homo sapiens | ? | - |
? | |
Phe-Gly + H2O | - |
Homo sapiens | Phe + Gly | - |
? | |
Trp-Gly + H2O | - |
Homo sapiens | Trp + Gly | - |
? | |
Val-Gly + H2O | - |
Homo sapiens | Val + Gly | - |
? |