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Literature summary for 3.4.11.18 extracted from

  • Warder, S.E.; Tucker, L.A.; McLoughlin, S.M.; Strelitzer, T.J.; Meuth, J.L.; Zhang, Q.; Sheppard, G.S.; Richardson, P.L.; Lesniewski, R.; Davidsen, S.K.; Bell, R.L.; Rogers, J.C.; Wang, J.
    Discovery, identification, and characterization of candidate pharmacodynamic markers of methionine aminopeptidase-2 inhibition (2008), J. Proteome Res., 7, 4807-4820.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
A-357300 potent MetAP2 inhibitor Homo sapiens
A-357300 potent MetAP2 inhibitor Mus musculus
A-800141 potent MetAP2 inhibitor Homo sapiens
A-800141 potent MetAP2 inhibitor Mus musculus
fumagillin potent MetAP2 inhibitor Homo sapiens
fumagillin potent MetAP2 inhibitor Mus musculus
TNP-470 potent MetAP2 inhibitor Homo sapiens
TNP-470 potent MetAP2 inhibitor Mus musculus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
Mono Q column chromatography and Q-Sepharose column chromatography Mus musculus
Mono Q column chromatography and Q-Sepharose column chromatography Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
erythroleukemia cell
-
Mus musculus
-
HT-1080 cell
-
Homo sapiens
-
K-562 cell
-
Homo sapiens
-
MEL cell
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
cyclophillin A + H2O MetAP2-specific substrate Mus musculus ?
-
?
cyclophillin A + H2O MetAP2-specific substrate Homo sapiens ?
-
?
eukaryotic elongation factor-2 + H2O MetAP2-specific substrate Mus musculus ?
-
?
eukaryotic elongation factor-2 + H2O MetAP2-specific substrate Homo sapiens ?
-
?
glyceraldehye 3-phosphate dehydrogenase + H2O MetAP2-specific substrate Mus musculus ?
-
?
glyceraldehye 3-phosphate dehydrogenase + H2O MetAP2-specific substrate Homo sapiens ?
-
?
L-Met-L-Pro-p-nitroanilide + H2O
-
Mus musculus L-Met + L-Pro-p-nitroanilide
-
?
L-Met-L-Pro-p-nitroanilide + H2O
-
Homo sapiens L-Met + L-Pro-p-nitroanilide
-
?
SH3 binding glutamic acid rich-like protein + H2O MetAP2-specific substrate Mus musculus ?
-
?
SH3 binding glutamic acid rich-like protein + H2O MetAP2-specific substrate Homo sapiens ?
-
?
thioredoxin-1 + H2O MetAP2-specific substrate Mus musculus ?
-
?
thioredoxin-1 + H2O MetAP2-specific substrate Homo sapiens ?
-
?

Synonyms

Synonyms Comment Organism
MetAP2
-
Mus musculus
MetAP2
-
Homo sapiens
methionine aminopeptidase-2
-
Mus musculus
methionine aminopeptidase-2
-
Homo sapiens