Cloned (Comment) | Organism |
---|---|
expressed in NIH-3T3 cells and NL20 cell line | Homo sapiens |
Protein Variants | Comment | Organism |
---|---|---|
H231N | enzymatically inactive | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
A-357300 | - |
Homo sapiens | |
A-800141 | - |
Homo sapiens | |
fumagillin | - |
Homo sapiens | |
TNP-470 | irreversible inhibitor | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P50579 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
breast carcinoma cell | - |
Homo sapiens | - |
Calu-6 cell | - |
Homo sapiens | - |
colonic cancer cell | - |
Homo sapiens | - |
DLD-1 cell | - |
Homo sapiens | - |
HCT-116 cell | - |
Homo sapiens | - |
HCT-15 cell | - |
Homo sapiens | - |
HT-1080 cell | - |
Homo sapiens | - |
LoVo cell | - |
Homo sapiens | - |
lung adenocarcinoma cell | - |
Homo sapiens | - |
NCI-H1299 cell | - |
Homo sapiens | - |
NCI-H460 cell | - |
Homo sapiens | - |
ovary cancer cell | - |
Homo sapiens | - |
PC-3 cell | - |
Homo sapiens | - |
prostate cancer cell | - |
Homo sapiens | - |
SW-620 cell | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
MetAP2 | - |
Homo sapiens |
methionine aminopeptidase-2 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000003 | - |
- |
Homo sapiens | TNP-470 | |
0.00002 | - |
- |
Homo sapiens | A-800141 | |
0.00015 | - |
- |
Homo sapiens | A-357300 |