Activating Compound | Comment | Organism | Structure |
---|---|---|---|
isoproterenol | 0.001 mM isoproterenol triggers a sustained, 2fold increase in PDE4 activity | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
rolipram | specific PDE4 inhibitor, complete inhibition at 0.01 mM rolipram | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HEK-293 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | - |
Homo sapiens | 5'-AMP | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PDE4 | - |
Homo sapiens |