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Literature summary for 3.1.4.53 extracted from

  • Xin, W.; Tran, T.M.; Richter, W.; Clark, R.B.; Rich, T.C.
    Roles of GRK and PDE4 activities in the regulation of beta2 adrenergic signaling (2008), J. Gen. Physiol., 131, 349-364.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
isoproterenol 0.001 mM isoproterenol triggers a sustained, 2fold increase in PDE4 activity Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
rolipram specific PDE4 inhibitor, complete inhibition at 0.01 mM rolipram Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
HEK-293 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3',5'-cAMP + H2O
-
Homo sapiens 5'-AMP
-
?

Synonyms

Synonyms Comment Organism
PDE4
-
Homo sapiens