Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(R)-rolipram | - |
Homo sapiens | |
denbufylline | - |
Homo sapiens | |
additional information | no inhibition by siguazodan or zaprinast | Homo sapiens | |
Ro20-1724 | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0043 | - |
adenosine 3',5'-cyclic phosphate | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q07343 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Homo sapiens | - |
frontal lobe | - |
Homo sapiens | - |
heart | - |
Homo sapiens | - |
lung | - |
Homo sapiens | - |
additional information | PDE IVB is not detected in Placenta, liver, kidney, or pancreas | Homo sapiens | - |
skeletal muscle | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
adenosine 3',5'-cyclic phosphate + H2O | - |
Homo sapiens | adenosine 5'-phosphate | - |
? | |
additional information | no hydrolysis of cGMP | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
cAMP-specific phosphodiesterase | - |
Homo sapiens |
PDE IVB | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000085 | - |
(R)-rolipram | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0005 | - |
- |
Homo sapiens | denbufylline | |
0.0022 | - |
- |
Homo sapiens | Ro20-1724 |