Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Leishmania major |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(2E)-9,10-dimethoxy-3-methyl-2-[(2,4,6-trimethylphenyl)imino]-2,3,6,7-tetrahydro-4H-pyrimido[6,1-a]isoquinolin-4-one | - |
Leishmania major | |
dipyridamole | - |
Leishmania major | |
etazolate | - |
Leishmania major | |
Milrinone | - |
Leishmania major | |
papaverine | - |
Leishmania major | |
rolipram | - |
Leishmania major |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00099 | - |
3',5'-cAMP | - |
Leishmania major | |
0.00698 | - |
3',5'-cAMP | - |
Leishmania major |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Leishmania major | Q6S996 | - |
- |
Leishmania major | Q6S997 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | LmjPDEB1 is completely cAMP-specific | Leishmania major | 5'-AMP | - |
? | |
3',5'-cAMP + H2O | LmjPDEB2 is completely cAMP-specific | Leishmania major | 5'-AMP | - |
? |
Synonyms | Comment | Organism |
---|---|---|
class I phosphodiesterase PDEB1 | - |
Leishmania major |
class I phosphodiesterase PDEB2 | - |
Leishmania major |
LmjPDEB1 | - |
Leishmania major |
LmjPDEB2 | - |
Leishmania major |