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Literature summary for 3.1.4.17 extracted from

  • Giorgi, M.; Caniglia, C.; Scarsella, G.; Augusti-Tocco, G.
    Characterization of 3':5' cyclic nucleotide phosphodiesterase activities of mouse neuroblastoma N18TG2 cells (1993), FEBS Lett., 324, 76-80.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
5-(2-propoxyphenyl)-2,3-dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
-
Mus musculus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information biphasic behaviour with 3',5'-cAMP as substrate Mus musculus
0.0088
-
3',5'-cGMP
-
Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
N18TG2 cell
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3',5'-cAMP + H2O
-
Mus musculus 5'-AMP
-
?
3',5'-cGMP + H2O
-
Mus musculus 5'-GMP
-
?

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0003
-
5-(2-propoxyphenyl)-2,3-dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidin-7-one
-
Mus musculus