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Literature summary for 3.1.4.11 extracted from

  • Shimizu, T.; Yamaguchi, N.; Okada, S.; Lu, L.; Sasaki, T.; Yokotani, K.
    Roles of brain phosphatidylinositol-specific phospholipase C and diacylglycerol lipase in centrally administered histamine-induced adrenomedullary outflow in rats (2007), Eur. J. Pharmacol., 571, 138-144.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
1-O-octadecyl-2-O-methyl-sn-glycero-3-phosphorylcholine histamine-induced elevation of plasma noradrenaline and adrenaline is dose-dependently reduced by ET-18-OCH3 Rattus norvegicus
additional information mepacrine (PLA2 inhibitor) and D609 (phosphatidylcholine-specific PLC inhibitor) have no effect. Histamine-induced elevation of plasma noradrenaline and adrenaline is also dose-dependently reduced by RHC-80267 (diacylglycerol lipase inhibitor) Rattus norvegicus
U-73122 histamine-induced elevation of plasma noradrenaline and adrenaline is dose-dependently reduced by U-73122 Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
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-
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Rattus norvegicus
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male Wistar rats
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Source Tissue

Source Tissue Comment Organism Textmining
blood plasma
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Rattus norvegicus
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brain
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Rattus norvegicus
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brain involvement of brain phosphatidylinositol-specific phospholipase C in the centrally administered histamine-induced activation of the adrenomedullary outflow in rats Rattus norvegicus
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Synonyms

Synonyms Comment Organism
phosphatidylinositol-specific phospholipase C
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Rattus norvegicus