Inhibitors | Comment | Organism | Structure |
---|---|---|---|
eserine | native enzyme, 50% inhibition at 5 nM, recombinant enzyme, 50% inhibition at 5 nM | Homo sapiens | |
ethyl carbamoyl | native enzyme, 50% inhibition at 10 nM, recombinant enzyme, 50% inhibition at 5 nM | Homo sapiens | |
phenethyl cymserine | native enzyme, 50% inhibition at 7 nM, recombinant enzyme, 50% inhibition at 50 nM | Homo sapiens | |
phenserine | native enzyme, 50% inhibition at 500 nM, recombinant enzyme, 50% inhibition at 500 nM | Homo sapiens | |
pyridostigmine bromide | native enzyme, 50% inhibition at 300 nM, recombinant enzyme, 50% inhibition at 500 nM | Homo sapiens | |
tolserine | native enzyme, 50% inhibition at 50 nM, recombinant enzyme, 50% inhibition at 80 nM | Homo sapiens | |
tolserine N-dimethyl ammonium bromide | native enzyme, 50% inhibition at 44 nM, recombinant enzyme, 50% inhibition at 45 nM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
native enzyme and recombinant enzyme expressed in milk of transgenic goat | - |
Source Tissue | Comment | Organism | Textmining |
---|
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00000088 | - |
eserine | 22°C | Homo sapiens | |
0.00000174 | - |
eserine | 22°C | Homo sapiens | |
0.0000071 | - |
ethyl carbamoyl | 22°C | Homo sapiens | |
0.0000152 | - |
phenethyl cymserine | 22°C | Homo sapiens | |
0.000023 | - |
ethyl carbamoyl | 22°C | Homo sapiens | |
0.0000356 | - |
phenethyl cymserine | 22°C | Homo sapiens | |
0.000073 | - |
tolserine | 22°C | Homo sapiens | |
0.00009 | - |
tolserine N-dimethyl ammonium bromide | 22°C | Homo sapiens | |
0.000139 | - |
tolserine | 22°C | Homo sapiens | |
0.00046 | - |
pyridostigmine bromide | 22°C | Homo sapiens | |
0.000616 | - |
pyridostigmine bromide | 22°C | Homo sapiens | |
0.000655 | - |
phenserine | 22°C | Homo sapiens | |
0.0013 | - |
phenserine | 22°C | Homo sapiens |