Application | Comment | Organism |
---|---|---|
diagnostics | the enzyme has potential as biomarker of pesticides and metal ions | Parachromis managuensis |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
BW284c51 | - |
Parachromis managuensis | |
Carbaryl | - |
Parachromis managuensis | |
carbofuran | - |
Parachromis managuensis | |
Cd2+ | 25% inhibition at 1 mM | Parachromis managuensis | |
Cu2+ | 53% inhibition at 1 mM | Parachromis managuensis | |
dichlorvos | - |
Parachromis managuensis | |
eserine | - |
Parachromis managuensis | |
Hg2+ | complete inhibition at 1 mM | Parachromis managuensis | |
iso-ompa | - |
Parachromis managuensis | |
Mn2+ | about 20% inhibition at 1 mM | Parachromis managuensis | |
neostigmine | - |
Parachromis managuensis | |
Pb2+ | slight inhibition | Parachromis managuensis | |
Zn2+ | 17% inhibition at 1 mM | Parachromis managuensis |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | Michaelis-Menten kinetics | Parachromis managuensis | |
0.59 | - |
acetylthiocholine | pH 8.0, 25°C | Parachromis managuensis |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
additional information | no or poor effect by Al3+, Ba2+, Mg2+, Mn2+, and Fe2+ at 1 mM | Parachromis managuensis |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylcholine + H2O | Parachromis managuensis | - |
choline + acetate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Parachromis managuensis | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Parachromis managuensis | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylcholine + H2O | - |
Parachromis managuensis | choline + acetate | - |
? | |
acetylthiocholine + H2O | - |
Parachromis managuensis | thiocholine + acetate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
AChE | - |
Parachromis managuensis |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
35 | - |
- |
Parachromis managuensis |
Temperature Minimum [°C] | Temperature Maximum [°C] | Comment | Organism |
---|---|---|---|
20 | 40 | over 60% of maximal activity within this range | Parachromis managuensis |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
- |
Parachromis managuensis |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
7 | 9 | over 60% of maximal activity within this range | Parachromis managuensis |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00012 | - |
Hg2+ | pH 8.0, 25°C | Parachromis managuensis | |
0.0012 | - |
eserine | pH 8.0, 25°C | Parachromis managuensis | |
0.0014 | - |
iso-ompa | pH 8.0, 25°C | Parachromis managuensis | |
0.0044 | - |
neostigmine | pH 8.0, 25°C | Parachromis managuensis | |
0.00725 | - |
Cu2+ | pH 8.0, 25°C | Parachromis managuensis | |
0.0082 | - |
BW284c51 | pH 8.0, 25°C | Parachromis managuensis | |
0.0343 | - |
Cd2+ | pH 8.0, 25°C | Parachromis managuensis | |
0.1216 | - |
Zn2+ | pH 8.0, 25°C | Parachromis managuensis |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.013 | - |
pH 8.0, 25°C | Parachromis managuensis | Hg2+ | |
0.1165 | - |
pH 8.0, 25°C | Parachromis managuensis | Zn2+ | |
0.17 | - |
pH 8.0, 25°C | Parachromis managuensis | eserine | |
0.2 | - |
pH 8.0, 25°C | Parachromis managuensis | iso-ompa | |
0.61 | - |
pH 8.0, 25°C | Parachromis managuensis | neostigmine | |
0.773 | - |
pH 8.0, 25°C | Parachromis managuensis | Cu2+ | |
0.87 | - |
pH 8.0, 25°C | Parachromis managuensis | BW284c51 | |
3.656 | - |
pH 8.0, 25°C | Parachromis managuensis | Cd2+ | |
7.75 | - |
pH 8.0, 25°C | Parachromis managuensis | Pb2+ | |
12.969 | - |
pH 8.0, 25°C | Parachromis managuensis | Zn2+ |