Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | poor inhibition of 0-2% by N,N,N-trimethyl-17-(methylsulfonylthio)heptadecan-1-aminium bromide, i.e. AMTS17, N,N,N-trimethyl-18-(methylsulfonylthio)octadecan-1-aminium bromide, i.e. AMTS18, N,N,N-trimethyl-19-(methylsulfonylthio)nonadecan-1-aminium bromide, i.e. AMTS19, and N,N,N-trimethyl-20-(methylsulfonylthio)eicosan-1-aminiumbromide, i.e. i.e. AMTS20 | Homo sapiens | |
N,N,N-trimethyl-10-(methylsulfonylthio)decan-1-aminium bromide | i.e. AMTS10, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-10-(methylsulfonylthio)decan-1-aminium bromide | i.e. AMTS10, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-11-(methylsulfonylthio)undecan-1-aminium bromide | i.e. AMTS11, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-11-(methylsulfonylthio)undecan-1-aminium bromide | i.e. AMTS11, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-12-(methylsulfonylthio)dodecan-1-aminium bromide | i.e. AMTS12, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-12-(methylsulfonylthio)dodecan-1-aminium bromide | i.e. AMTS12, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-13-(methylsulfonylthio)tridecan-1-aminium bromide | i.e. AMTS13, causes a degree of apparently irreversible of the AChE activity in erythrocytes. AMTS13 at 0.006 mM leads to 43% inhibition after 1 h, 70% after 6 h, and 78% after 16 h | Homo sapiens | |
N,N,N-trimethyl-13-(methylsulfonylthio)tridecan-1-aminium bromide | i.e. AMTS13, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-14-(methylsulfonylthio)tetradecan-1-aminium bromide | i.e. AMTS14, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-14-(methylsulfonylthio)tetradecan-1-aminium bromide | i.e. AMTS14, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-15-(methylsulfonylthio)pentadecan-1-aminium bromide | i.e. AMTS15, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-15-(methylsulfonylthio)pentadecan-1-aminium bromide | i.e. AMTS15, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-16-(methylsulfonylthio)hexadecan-1-aminium bromide | i.e. AMTS16, causes a degree of apparently irreversible of the AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-16-(methylsulfonylthio)hexadecan-1-aminium bromide | i.e. AMTS16, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-17-(methylsulfonylthio)heptadecan-1-aminium bromide | i.e. AMTS17, irreversibly inhibits 99% of the AChE activity in greenbug extracts, AChE species-selectivity | Schizaphis graminum | |
N,N,N-trimethyl-18-(methylsulfonylthio)octadecan-1-aminium bromide | i.e. AMTS18, irreversibly inhibits 99% of the AChE activity in greenbug extracts, AChE species-selectivity | Schizaphis graminum | |
N,N,N-trimethyl-19-(methylsulfonylthio)nonadecan-1-aminium bromide | i.e. AMTS19, irreversibly inhibits 99% of the AChE activity in greenbug extracts, AChE species-selectivity | Schizaphis graminum | |
N,N,N-trimethyl-20-(methylsulfonylthio)eicosan-1-aminiumbromi de | i.e. AMTS20, irreversibly inhibits 99% of the AChE activity in greenbug extracts, AChE species-selectivity | Schizaphis graminum | |
N,N,N-trimethyl-7-(methylsulfonylthio)heptan-1-aminium bromide | i.e. AMTS7, causes weak and purely reversible inhibition of AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-7-(methylsulfonylthio)heptan-1-aminium bromide | i.e. AMTS7, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-8-(methylsulfonylthio)octan-1-aminium bromide | i.e. AMTS8, causes weak and purely reversible inhibition of AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-8-(methylsulfonylthio)octan-1-aminium bromide | i.e. AMTS8, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum | |
N,N,N-trimethyl-9-(methylsulfonylthio)nonan-1-aminium bromide | i.e. AMTS9, causes weak and purely reversible inhibition of AChE activity in erythrocytes | Homo sapiens | |
N,N,N-trimethyl-9-(methylsulfonylthio)nonan-1-aminium bromide | i.e. AMTS9, irreversibly inhibits over 87% of the AChE activity in greenbug extracts | Schizaphis graminum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Schizaphis graminum | - |
greenbug aphid | - |
Purification (Comment) | Organism |
---|---|
native enzyme from greenbug aphids | Homo sapiens |
native enzyme from greenbug aphids | Schizaphis graminum |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
erythrocyte | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
AChE | - |
Homo sapiens |
AChE | - |
Schizaphis graminum |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
37 | - |
assay at | Schizaphis graminum |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Homo sapiens |
7.4 | - |
assay at | Schizaphis graminum |