Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Ethidium bromide | uncompetitive inhibition at concentrations of 0.00625-0.1 mM in all brain regions except for the cerebellum where the inhibition is of a mixed-type | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Rattus norvegicus | - |
cerebellum | - |
Rattus norvegicus | - |
cerebral cortex | - |
Rattus norvegicus | - |
hippocampus | - |
Rattus norvegicus | - |
striatum | - |
Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylthiocholine + H2O | - |
Rattus norvegicus | thiocholine + acetate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
AChE | - |
Rattus norvegicus |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | - |
assay at | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
assay at | Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | tissue-dependent inhibition kinetics, overview | Rattus norvegicus | |
0.0024 | 0.0059 | Ethidium bromide | pH 7.5, 25°C | Rattus norvegicus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0049 | 0.009 | pH 7.5, 25°C | Rattus norvegicus | Ethidium bromide |