Inhibitors | Comment | Organism | Structure |
---|---|---|---|
13beta,19-dihydroy-3,15-dioxoatis-16-ene-19-O-beta-D-(6'-galloyl)-glucopyranoside | - |
Homo sapiens | |
13beta,19-dihydroy-3,15-dioxoatis-16-ene-19-O-beta-Dglucopyranoside | - |
Homo sapiens | |
4beta,9alpha,16,20-tetrahydroxy-14(13->12)-abeo-12alphaH-1,6-tigliadiene-3,13-dione | competitive inhibition | Homo sapiens | |
4beta,9alpha,20-trihydroxy-14(13->12)-abeo-12alphaH-1,6-tigliadiene-3,13-dione | - |
Homo sapiens | |
bisdehydrophorbol | - |
Homo sapiens | |
didehydrolangduin A-20-O-beta-D-glucopyranoside | - |
Homo sapiens | |
ent-16beta,17-dihydroxyatisan-3-one-19-O-beta-D-(6'-galloyl)-glucopyranoside | - |
Homo sapiens | |
ent-16beta,17-dihydroxyatisan-3-one-19-O-beta-D-glucopyranoside | - |
Homo sapiens | |
ent-kaurane-16beta,17-diol-3,12-dione-19-O-beta-D-glucopyranoside | - |
Homo sapiens | |
ent-kaurane-16beta,17-diol-3-one-19-O-beta-D-(6'-galloyl)-glucopyranoside | - |
Homo sapiens | |
ent-kaurane-16beta,17-diol-3-one-19-O-beta-D-glucopyranoside | - |
Homo sapiens | |
fischeroside A | - |
Homo sapiens | |
fischeroside A-16-O-beta-D-glucopyranoside | - |
Homo sapiens | |
ingenol-19-O-beta-D-glucopyranoside | - |
Homo sapiens | |
langduin F | - |
Homo sapiens | |
additional information | diterpenoids and glycosides are isolated from roots of Euphorbia ebracteolata and their inhibitory potency and structure is determined, NMR spectrometric analysis, overview | Homo sapiens | |
phorbol-13-acetate | - |
Homo sapiens | |
yuexiandajisu D | - |
Homo sapiens | |
yuexiandajisu E | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | O00748 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
intestine | - |
Homo sapiens | - |
liver | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
carboxylesterase 2 | - |
Homo sapiens |
hCE-2 | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00494 | - |
4beta,9alpha,16,20-tetrahydroxy-14(13->12)-abeo-12alphaH-1,6-tigliadiene-3,13-dione | pH and temperature not specified in the publication | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00388 | - |
pH and temperature not specified in the publication | Homo sapiens | 4beta,9alpha,16,20-tetrahydroxy-14(13->12)-abeo-12alphaH-1,6-tigliadiene-3,13-dione | |
0.00395 | - |
pH and temperature not specified in the publication | Homo sapiens | 4beta,9alpha,20-trihydroxy-14(13->12)-abeo-12alphaH-1,6-tigliadiene-3,13-dione | |
0.00447 | - |
pH and temperature not specified in the publication | Homo sapiens | yuexiandajisu E | |
0.00479 | - |
pH and temperature not specified in the publication | Homo sapiens | yuexiandajisu D | |
0.00499 | - |
pH and temperature not specified in the publication | Homo sapiens | bisdehydrophorbol | |
0.00521 | - |
pH and temperature not specified in the publication | Homo sapiens | langduin F | |
0.00883 | - |
pH and temperature not specified in the publication | Homo sapiens | phorbol-13-acetate | |
0.01346 | - |
pH and temperature not specified in the publication | Homo sapiens | didehydrolangduin A-20-O-beta-D-glucopyranoside | |
0.01786 | - |
pH and temperature not specified in the publication | Homo sapiens | ent-16beta,17-dihydroxyatisan-3-one-19-O-beta-D-(6'-galloyl)-glucopyranoside | |
0.02168 | - |
pH and temperature not specified in the publication | Homo sapiens | fischeroside A | |
0.0293 | - |
pH and temperature not specified in the publication | Homo sapiens | fischeroside A-16-O-beta-D-glucopyranoside | |
0.03249 | - |
pH and temperature not specified in the publication | Homo sapiens | ingenol-19-O-beta-D-glucopyranoside | |
0.05327 | - |
pH and temperature not specified in the publication | Homo sapiens | ent-kaurane-16beta,17-diol-3-one-19-O-beta-D-(6'-galloyl)-glucopyranoside | |
0.1 | - |
pH and temperature not specified in the publication | Homo sapiens | 13beta,19-dihydroy-3,15-dioxoatis-16-ene-19-O-beta-D-(6'-galloyl)-glucopyranoside | |
0.1 | - |
pH and temperature not specified in the publication | Homo sapiens | 13beta,19-dihydroy-3,15-dioxoatis-16-ene-19-O-beta-Dglucopyranoside | |
0.1 | - |
pH and temperature not specified in the publication | Homo sapiens | ent-16beta,17-dihydroxyatisan-3-one-19-O-beta-D-glucopyranoside | |
0.1 | - |
pH and temperature not specified in the publication | Homo sapiens | ent-kaurane-16beta,17-diol-3,12-dione-19-O-beta-D-glucopyranoside | |
0.1 | - |
pH and temperature not specified in the publication | Homo sapiens | ent-kaurane-16beta,17-diol-3-one-19-O-beta-D-glucopyranoside |
General Information | Comment | Organism |
---|---|---|
evolution | the enzyme belongs to the serine protease superfamily | Homo sapiens |