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Literature summary for 2.7.7.49 extracted from

  • Held, D.M.; Kissel, J.D.; Saran, D.; Michalowski, D.; Burke, D.H.
    Differential susceptibility of HIV-1 reverse transcriptase to inhibition by RNA aptamers in enzymatic reactions monitoring specific steps during genome replication (2006), J. Biol. Chem., 281, 25712-25722.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
2',3'-dideoxy-CTP
-
Human immunodeficiency virus 1
azidothymidine triphosphate
-
Human immunodeficiency virus 1
efavirenz
-
Human immunodeficiency virus 1
nevirapine
-
Human immunodeficiency virus 1
RNA aptamer RNA aptamers suppress viral replication by cumulative inhibition of reverse transcriptase at every stage of genome replication Human immunodeficiency virus 1

Localization

Localization Comment Organism GeneOntology No. Textmining

Organism

Organism UniProt Comment Textmining
Human immunodeficiency virus 1
-
-
-

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
additional information
-
IC50-values of aptamers Human immunodeficiency virus 1 additional information
0.00006
-
-
Human immunodeficiency virus 1 efavirenz
0.00129
-
-
Human immunodeficiency virus 1 nevirapine
0.00134
-
-
Human immunodeficiency virus 1 azidothymidine triphosphate
0.00224
-
-
Human immunodeficiency virus 1 2',3'-dideoxy-CTP