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BRENDA support

Literature summary for 2.7.11.18 extracted from

  • Luh, C.; Kuhlmann, C.R.; Ackermann, B.; Timaru-Kast, R.; Luhmann, H.J.; Behl, C.; Werner, C.; Engelhard, K.; Thal, S.C.
    Inhibition of myosin light chain kinase reduces brain edema formation after traumatic brain injury (2009), J. Neurochem., 112, 1015-1025.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
ML-7 selective MLCK inhibitor Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + myosin light chain
-
Mus musculus ADP + myosin light chain phosphate
-
?

Synonyms

Synonyms Comment Organism
MLCK
-
Mus musculus
myosin light chain kinase
-
Mus musculus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Mus musculus

Expression

Organism Comment Expression
Mus musculus MLCK expression is significantly up-regulated after controlled cortical impact with a maximum 12 h post-injury up

General Information

General Information Comment Organism
physiological function phosphorylation of myosin light chains by myosin light chain kinase activates endothelial contractile elements and results in a rearrangement of the cytoskeleton Mus musculus