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Literature summary for 2.7.11.17 extracted from

  • Kemp, B.E.; Parker, M.W.; Hu, S.; Tiganis, T.; House, C.
    Substrate and pseudosubstrate interactions with protein kinases: determinants of specificity (1994), Trends Biochem. Sci., 19, 440-444.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information autoregulation by a pseudosubstrate mechanism, overview Mammalia

Inhibitors

Inhibitors Comment Organism Structure
additional information the enzyme is inhibited by its regulatory subunit masking the active site, autoregulation by a pseudosubstrate mechanism, overview Mammalia

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ binding required for activity Mammalia

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + a protein Mammalia
-
ADP + a phosphoprotein
-
?

Organism

Organism UniProt Comment Textmining
Mammalia
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + a protein
-
Mammalia ADP + a phosphoprotein
-
?
additional information substrate specificity and binding structure, the enzyme depends on basic residues for substrate recognition, autoregulation by a pseudosubstrate mechanism, overview Mammalia ?
-
?

Synonyms

Synonyms Comment Organism
CaMKII
-
Mammalia

Cofactor

Cofactor Comment Organism Structure
ATP
-
Mammalia
Calmodulin binding required for activity Mammalia