Cloned (Comment) | Organism |
---|---|
beta-ARK 1 is cloned and expressed in SF9 cells using the baculovirus expression system | Homo sapiens |
beta-ARK 1 is cloned and expressed in SF9 cells using the baculovirus expression system | Bos taurus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0038 | - |
rhodopsin | pH 7.5, 30°C, recombinant beta-ARK 1 | Bos taurus | |
0.022 | - |
ATP | pH 7.5, 30°C, recombinant beta-ARK 1, rhodopsin as substrate | Bos taurus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | - |
Homo sapiens | 5829 | - |
cytosol | - |
Bos taurus | 5829 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | requirement | Homo sapiens | |
Mg2+ | requirement | Bos taurus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + beta-adrenergic receptor | Homo sapiens | natural substrate: beta2-adrenergic receptor | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | Bos taurus | natural substrate: beta2-adrenergic receptor | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | Homo sapiens | agonist-occupied form of the receptor | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | Bos taurus | agonist-occupied form of the receptor | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | Homo sapiens | involved in homologous desensitization of beta-adrenergic receptor | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | Bos taurus | involved in homologous desensitization of beta-adrenergic receptor | ADP + phospho-beta-adrenergic receptor | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
enzyme exists in 2 subtypes: beta-ARK 1 and beta-ARK 2 | - |
Bos taurus | - |
major isoform beta-ARK 1 | - |
Homo sapiens | - |
major isoform beta-ARK 1 | - |
Homo sapiens | - |
enzyme exists in 2 subtypes: beta-ARK1 and 2 | - |
Purification (Comment) | Organism |
---|---|
recombinant beta-ARK 1 expressed in Sf9 cells | Bos taurus |
recombinant beta-ARK 1, expressed in Sf9 cells | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Bos taurus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + beta-adrenergic receptor | specifically phosphorylates the agonist-occupied form of the receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | specifically phosphorylates the agonist-occupied form of the receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | human beta2-adrenergic receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | human beta2-adrenergic receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | incorporation of up to 5 mol phosphate/mol receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | incorporation of up to 5 mol phosphate/mol receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | beta-AR from Sf9 cells | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | beta-AR from Sf9 cells | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | natural substrate: beta2-adrenergic receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | natural substrate: beta2-adrenergic receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | agonist-occupied form of the receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | agonist-occupied form of the receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | involved in homologous desensitization of beta-adrenergic receptor | Homo sapiens | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + beta-adrenergic receptor | involved in homologous desensitization of beta-adrenergic receptor | Bos taurus | ADP + phospho-beta-adrenergic receptor | - |
? | |
ATP + rhodopsin | in form of bovine rod outer segments | Homo sapiens | ADP + phosphorhodopsin | - |
? | |
ATP + rhodopsin | in form of bovine rod outer segments | Bos taurus | ADP + phosphorhodopsin | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
30 | - |
assay at | Homo sapiens |
30 | - |
assay at | Bos taurus |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
ATP | - |
Bos taurus | |
ATP | cofactor ATP | Homo sapiens |