Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 2.7.11.11 extracted from

  • Dai, R.; Ali, M.K.; Lezcano, N.; Bergson, C.
    A crucial role for cAMP and protein kinase A in D1 dopamine receptor regulated intracellular calcium transients (2008), Neurosignals, 16, 112-123.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
8-bromo-cAMP 1 mM Homo sapiens
8-bromo-cAMP 1 mM Rattus norvegicus
forskolin 0.01 mM Homo sapiens
forskolin 0.01 mM Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
H-89
-
Homo sapiens
H-89
-
Rattus norvegicus
KT-5720
-
Homo sapiens
KT-5720
-
Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
D1-HEK-293 cell HEK-293 cells that stably express D1 receptors Homo sapiens
-
hippocampus
-
Rattus norvegicus
-
neuron
-
Rattus norvegicus
-

Synonyms

Synonyms Comment Organism
PKA
-
Homo sapiens
PKA
-
Rattus norvegicus
protein kinase A
-
Homo sapiens
protein kinase A
-
Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens
ATP
-
Rattus norvegicus
cAMP dependent Homo sapiens
cAMP dependent Rattus norvegicus