Application | Comment | Organism |
---|---|---|
medicine | inhibition of IkappaB kinase beta restrains oncogenic proliferation of pancreatic cancer cells | Mus musculus |
medicine | inhibition of IkappaB kinase beta restrains oncogenic proliferation of pancreatic cancer cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
IMD-0354 | specific IKKbeta inhibition | Homo sapiens | |
IMD-0354 | specific IKKbeta inhibition | Mus musculus | |
RNAi | specific IKKbeta inhibition | Homo sapiens | |
RNAi | specific IKKbeta inhibition | Mus musculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + [IkappaB protein] | Mus musculus | - |
ADP + [IkappaB phosphoprotein] | - |
? | |
ATP + [IkappaB protein] | Homo sapiens | - |
ADP + [IkappaB phosphoprotein] | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
PANC-1 cell | - |
Homo sapiens | - |
pancreas | - |
Mus musculus | - |
PK-8 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + [IkappaB protein] | - |
Mus musculus | ADP + [IkappaB phosphoprotein] | - |
? | |
ATP + [IkappaB protein] | - |
Homo sapiens | ADP + [IkappaB phosphoprotein] | - |
? |
Synonyms | Comment | Organism |
---|---|---|
IkappaB kinase beta | - |
Mus musculus |
IkappaB kinase beta | - |
Homo sapiens |
IKKbeta | - |
Mus musculus |
IKKbeta | - |
Homo sapiens |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
ATP | - |
Mus musculus | |
ATP | - |
Homo sapiens |
General Information | Comment | Organism |
---|---|---|
physiological function | IkappaB kinase is a central kinase for nuclear factor-kappaB activation | Mus musculus |
physiological function | IkappaB kinase is a central kinase for nuclear factor-kappaB activation | Homo sapiens |