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BRENDA support

Literature summary for 2.7.10.2 extracted from

  • MacPartlin, M.; Smith, A.M.; Druker, B.J.; Honigberg, L.A.; Deininger, M.W.
    Brutons tyrosine kinase is not essential for Bcr-Abl-mediated transformation of lymphoid or myeloid cells (2008), Leukemia, 22, 1354-1360.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
LFM-A13
-
Mus musculus
PC-005
-
Mus musculus
PCI-31523
-
Mus musculus
shRNA
-
Mus musculus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + [protein]-L-tyrosine Mus musculus
-
ADP + [protein]-L-tyrosine phosphate
-
?

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Posttranslational Modification

Posttranslational Modification Comment Organism
phosphoprotein
-
Mus musculus

Source Tissue

Source Tissue Comment Organism Textmining
32D cell
-
Mus musculus
-
BA/F3 cell
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + [protein]-L-tyrosine
-
Mus musculus ADP + [protein]-L-tyrosine phosphate
-
?

Synonyms

Synonyms Comment Organism
Bruton's tyrosine kinase
-
Mus musculus
Btk
-
Mus musculus

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0000172
-
-
Mus musculus LFM-A13