Inhibitors | Comment | Organism | Structure |
---|---|---|---|
afatinib | - |
Homo sapiens | |
AG1478 | - |
Homo sapiens | |
cabozantinib | - |
Homo sapiens | |
cetuximab | - |
Homo sapiens | |
dacomitinib | - |
Homo sapiens | |
erlotinib | - |
Homo sapiens | |
foretinib | - |
Homo sapiens | |
gefitinib | - |
Homo sapiens | |
Genentech 5D5Fab | - |
Homo sapiens | |
lapatinib | - |
Homo sapiens | |
PHA-665752 | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a [protein]-L-tyrosine | Homo sapiens | - |
ADP + a [protein]-L-tyrosine phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
PC-3 cell | - |
Homo sapiens | - |
prostate adenocarcinoma cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a [protein]-L-tyrosine | - |
Homo sapiens | ADP + a [protein]-L-tyrosine phosphate | - |
? | |
ATP + poly-Ala-Glu-Lys-Tyr | substrate used for c-Met | Homo sapiens | ADP * poly-Ala-L-Glu-L-Lys-L-tyrosine phosphate | - |
? | |
ATP + poly-Glu-Tyr | substrate used for EGFR | Homo sapiens | ADP + poly-L-Glu-L-tyrosine phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
c-met | - |
Homo sapiens |
Egfr | - |
Homo sapiens |