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Literature summary for 2.7.1.40 extracted from

  • Derks, T.G.; van Dijk, T.H.; Grefhorst, A.; Rake, J.; Smit, G.P.; Kuipers, F.; Reijngoud, D.
    Inhibition of mitochondrial fatty acid oxidation in vivo only slightly suppresses gluconeogenesis but enhances clearance of glucose in mice (2008), Hepatology, 47, 1032-1042.
    View publication on PubMed

Application

Application Comment Organism
medicine acute pharmacological inhibiton of mitochondrial fatty acid oxidation using 2-tetradecylglcidic acid has no effect on endogenous glucose production and only a marginal effect on de novo glucose 6-phosphate synthesis Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
2-tetradecylglycidic acid in mice treated with 2-tetradecylglycidic acid, hepatic pyruvate kinase mRNA levels are significantly decreased, whereas pyruvate dehydrogenase kinase isozyme 4 expression is 30fold increased Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
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