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Literature summary for 2.7.1.32 extracted from

  • Rodriguez-Gonzalez, A.; Ramirez de Molina, A.; Banez-Coronel, M.; Megias, D.; Lacal, J.C.
    Inhibition of choline kinase renders a highly selective cytotoxic effect in tumour cells through a mitochondrial independent mechanism (2005), Int. J. Oncol., 26, 999-1008.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
MN58b specific inhibitor, IC50: 0.0005-0.072 mM depending on cell type Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
breast adenocarcinoma cell
-
Homo sapiens
-
cervical adenocarcinoma cell
-
Homo sapiens
-
colonic adenocarcinoma cell
-
Homo sapiens
-
epidermoid carcinoma cell
-
Homo sapiens
-
erythroleukemia cell
-
Homo sapiens
-
fibroblast
-
Homo sapiens
-
lymphoma cell
-
Homo sapiens
-
mammary epithelium
-
Homo sapiens
-
myeloma cell
-
Homo sapiens
-
osteosarcoma cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + choline
-
Homo sapiens ADP + O-phosphocholine
-
?

Synonyms

Synonyms Comment Organism
ChoK
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0005 0.072 specific inhibitor, IC50: 0.0005-0.072 mM depending on cell type Homo sapiens MN58b