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Literature summary for 2.7.1.153 extracted from

  • Vanhaesebroeck, B.; Welham, M.J.; Kotani, K.; Stein, R.; Warne, P.H.; Zvelebil, M.J.; Higashi, K.; Volinia, S.; Downward, J.; Waterfield, M.D.
    P110delta, a novel phosphoinositide 3-kinase in leukocytes (1997), Proc. Natl. Acad. Sci. USA, 94, 4330-4335.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
LY294002
-
Homo sapiens
Wortmannin
-
Homo sapiens

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
119471
-
x * 119471, p110delta subunit, can bind the p85 adaptor subunit, calculation from nucleotide sequence Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens O00329
-
-

Source Tissue

Source Tissue Comment Organism Textmining
leukocyte p110delta is exclusively localized in leukocytes Homo sapiens
-
MCF-7 cell
-
Homo sapiens
-
MOLT-4 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + 1-phosphatidyl-1D-myo-inositol 4,5-bisphosphate
-
Homo sapiens ADP + 1-phosphatidyl-1D-myo-inositol 3,4,5-trisphosphate
-
?
ATP + phosphatidylinositol
-
Homo sapiens ADP + phosphatidylinositol 3-phosphate
-
?
ATP + phosphatidylinositol 4-phosphate
-
Homo sapiens ADP + phosphatidylinositol 4,5-diphosphate
-
?
additional information p110delta does not phosphorylate the p85 adaptor but instead harbors an intrinsic autophosphorylation capacity Homo sapiens ?
-
?

Subunits

Subunits Comment Organism
? x * 119471, p110delta subunit, can bind the p85 adaptor subunit, calculation from nucleotide sequence Homo sapiens