Cloned (Comment) | Organism |
---|---|
class II phosphoinositide 3-kinase with a C2 domain, cloned from a U937 monocyte cDNA library, expression in mammalian and insect cells | Homo sapiens |
class II phosphoinositide 3-kinase, PI 3-kinase C2b, with a C2 domain is cloned from a U937 monocyte cDNA library and expressed in mammalian and insect cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Wortmannin | at nanomolar levels | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | can use either MgATP2- or CaATP2- | Homo sapiens | |
Mg2+ | can use either MgATP2- or CaATP2- | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
class II phosphoinositide 3-kinase, PI 3-kinase C2b | - |
Homo sapiens | O00750 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
cell culture | U937 monocyte | Homo sapiens | - |
cell culture | U937 monocytes | Homo sapiens | - |
monocyte | - |
Homo sapiens | - |
monocyte | U937 monocyte | Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + 1-phosphatidylinositol | - |
Homo sapiens | ADP + phosphatidylinositol 3-phosphate | - |
? | |
ATP + phosphatidylinositol 4,5-bisphosphate | no activity | Homo sapiens | ADP + phosphatidylinositol 3,4,5-trisphosphate | - |
? | |
ATP + phosphatidylinositol 4-phosphate | - |
Homo sapiens | ADP + phosphatidylinositol 3,4-bisphosphate | - |
? |