Activating Compound | Comment | Organism | Structure |
---|---|---|---|
additional information | not affected by 2,6-diaminopurine, 4-carbamoylimidazolium 5-olate, 8-azaadenine, and 2-fluoro-6-aminopurine | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
AMP | competitive against 5-phospho-alpha-D-ribose 1-diphosphate | Mus musculus | |
additional information | not affected by 2,6-diaminopurine, 4-carbamoylimidazolium 5-olate, 8-azaadenine, and 2-fluoro-6-aminopurine | Mus musculus | |
p-chloromercuribenzoate | no inhibition | Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0012 | - |
5-phospho-alpha-D-ribose 1-diphosphate | - |
Mus musculus | |
0.007 | - |
adenine | - |
Mus musculus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | required | Mus musculus | |
Mg2+ | absolute requirement | Mus musculus | |
Mg2+ | half-maximal activation at 0.4 mM | Mus musculus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
23000 | - |
2 * 23000, SDS-PAGE | Mus musculus |
44000 | - |
gel filtration | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Mus musculus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
F28-7 cell | cell line derived from FM3A | Mus musculus | - |
FM3A cell | mammary carcinoma cell line | Mus musculus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
20.6 | - |
purified enzyme | Mus musculus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
4-carbamoylimidazolium 5-olate + 5-phospho-alpha-D-ribose 1-diphosphate | low activity | Mus musculus | 4-carbamoylimidazolium 5-olate 5'-phosphate + diphosphate | - |
? | |
adenine + 5-phospho-alpha-D-ribose 1-diphosphate | - |
Mus musculus | AMP + diphosphate | - |
? |
Subunits | Comment | Organism |
---|---|---|
dimer | 2 * 23000, SDS-PAGE | Mus musculus |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
30 | - |
assay at | Mus musculus |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
7 | 9 | active over a broad range increasing progressively in activity from pH 7.0-9.0 | Mus musculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.024 | - |
AMP | - |
Mus musculus |