Inhibitors | Comment | Organism | Structure |
---|---|---|---|
benzimidazole | - |
Carica papaya | |
benzimidazole | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.019 | - |
glucagon(3-29) | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
0.087 | - |
Gln(3)-amyloid-beta peptide 3-11 amide | pH 6.0, 30°C, in absence of DMSO | Homo sapiens | |
0.089 | - |
Gln(3)-amyloid-beta peptide 3-40 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
0.155 | - |
Gln(3)-amyloid-beta peptide 3-11 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
0.162 | - |
Gln(3)-amyloid-beta peptide 3-21 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Carica papaya | - |
- |
- |
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Gln(3)-amyloid-beta peptide 3-11 amide | - |
Homo sapiens | ? | - |
? | |
Gln(3)-amyloid-beta peptide 3-21 amide | - |
Homo sapiens | ? | - |
? | |
Gln(3)-amyloid-beta peptide 3-40 amide | - |
Homo sapiens | ? | - |
? | |
Gln-2-naphthylamide | - |
Carica papaya | pyroglutamyl-2-naphthylamide + NH3 | - |
? | |
Glu-2-naphthylamide | - |
Carica papaya | ? | - |
? | |
glucagon(3-29) | - |
Homo sapiens | ? | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
10 | - |
glucagon(3-29) | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
40 | - |
Gln(3)-amyloid-beta peptide 3-40 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
41.4 | - |
Gln(3)-amyloid-beta peptide 3-11 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens | |
55 | - |
Gln(3)-amyloid-beta peptide 3-11 amide | pH 6.0, 30°C, in absence of DMSO | Homo sapiens | |
62 | - |
Gln(3)-amyloid-beta peptide 3-21 amide | pH 6.0, 30°C, 1% DMSO | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
6 | - |
cyclization of glutamic acid | Carica papaya |
8 | - |
cyclization of glutamine | Carica papaya |