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Literature summary for 2.3.1.26 extracted from

  • Chen, L.; Lafond, J.; Pelletier, R.M.
    A novel technical approach for the measurement of individual ACAT-1 and ACAT-2 enzymatic activity in the testis (2009), Methods Mol. Biol., 550, 169-177.
    View publication on PubMed

Application

Application Comment Organism
analysis use of inhibitor K-604, selective for isoform ACAT-1, to measure the individual enzymatic activities of isoforms ACAT-1 and ACAT-2 in semniferous tubule Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
K-604 selective for isoform ACAT-1, use to measure the individual enzymatic activities of isoforms ACAT-1 and ACAT-2; selective for isoform ACAT-1, use to measure the individual enzymatic activities of isoforms ACAT-1 and ACAT-2 Mus musculus
manassantin B inhibition of both isoforms ACAT-1 and ACAT-2; inhibition of both isoforms ACAT-1 and ACAT-2 Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus O88908 isoform ACAT2
-
Mus musculus Q61263 isoform ACAT1
-

Source Tissue

Source Tissue Comment Organism Textmining
seminiferous tubule
-
Mus musculus
-
testis
-
Mus musculus
-

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.1
-
isoform ACAT-1, semniferous tubules Mus musculus K-604
1
-
isoform ACAT-2, semniferous tubules Mus musculus K-604