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Literature summary for 2.1.1.28 extracted from

  • Kang, D.I.; Lee, J.Y.; Kim, W.; Jeong, K.W.; Shin, S.; Yang, J.; Park, E.; Chae, Y.K.; Kim, Y.
    Discovery of novel human phenylethanolamine N-methyltransferase (hPNMT) inhibitors using 3D pharmacophore-based in silico, biophysical screening and enzymatic activity assays (2010), Mol. Cells, 29, 595-602.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
expressed in Escherichia coli as a His-tagged fusion protein Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
1,4-diaminonaphthalene-2,6-disulfonic acid
-
Homo sapiens
4-(benzo[d][1,3]dioxol-5-ylamino)-4-oxobutanoic acid
-
Homo sapiens
4-oxo-1,4-dihydroquinoline-3,7-dicarboxylic acid
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
using Ni-NTA chromatography Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
S-adenosyl-L-methionine + noradrenaline
-
Homo sapiens S-adenosyl-L-homocysteine + epinephrine
-
?

Synonyms

Synonyms Comment Organism
hPNMT
-
Homo sapiens

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Homo sapiens