Activating Compound | Comment | Organism | Structure |
---|---|---|---|
ADP | ADP can reverse inhibition | Bos taurus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3,3'-[(2-bromobenzene-1,4-diyl)di(E)ethene-2,1-diyl]bis(6-hydroxybenzoic acid) | i.e. BSB | Bos taurus | |
ATP/GTP-competitive inhibitor of casein kinase-2 | - |
Bos taurus | |
aurintricarboxylic acid | - |
Bos taurus | |
BH3I-2 | - |
Bos taurus | |
bithionol | - |
Bos taurus | |
Calmidazolium | - |
Bos taurus | |
diethylstilbestrol | - |
Bos taurus | |
epicatechin | - |
Bos taurus | |
epicatechin-3-monogallate | - |
Bos taurus | |
epicatechin-monogallate | - |
Bos taurus | |
epigallocatechin | - |
Bos taurus | |
epigallocatechin-3,5-digallate | - |
Bos taurus | |
epigallocatechin-3-gallate | - |
Bos taurus | |
erythrosin B | - |
Bos taurus | |
ethaverine hydrochloride | - |
Bos taurus | |
gallic acid | - |
Bos taurus | |
GW-5074 | - |
Bos taurus | |
Hexachlorophene | - |
Bos taurus | |
leoidin | - |
Bos taurus | |
metergoline | - |
Bos taurus | |
suloctidil | - |
Bos taurus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
mitochondrion | - |
Bos taurus | 5739 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-glutamate + H2O + NAD+ | - |
Bos taurus | 2-oxoglutarate + NH3 + NADH + H+ | - |
? |
Synonyms | Comment | Organism |
---|---|---|
GDH | - |
Bos taurus |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
NAD+ | - |
Bos taurus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0005 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | epicatechin-3-monogallate | |
0.0005 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | epigallocatechin-3-monogallate | |
0.0012 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | aurintricarboxylic acid | |
0.0015 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | GW-5074 | |
0.0017 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | diethylstilbestrol | |
0.0017 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | Hexachlorophene | |
0.0037 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | BH3I-2 | |
0.0055 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | bithionol | |
0.0064 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | 3,3'-[(2-bromobenzene-1,4-diyl)di(E)ethene-2,1-diyl]bis(6-hydroxybenzoic acid) | |
0.0077 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | Calmidazolium | |
0.0138 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | suloctidil | |
0.0158 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | ATP/GTP-competitive inhibitor of casein kinase-2 | |
0.0328 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | metergoline | |
0.05 | - |
IC50 above 0.05 mM, in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | erythrosin B | |
0.08 | - |
in 0.1 M sodium phosphate buffer, pH 8.0, using 50 mM sodium glutamate and 0.2 mM NAD+ | Bos taurus | gallic acid |