Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3,4-dihydroxybenzoate | - |
Homo sapiens | |
ciclopirox olamine | - |
Homo sapiens | |
cobalt chloride | - |
Homo sapiens | |
Cu2+ | - |
Homo sapiens | |
deferoxamine | - |
Homo sapiens | |
dimethyloxalylglycine | - |
Homo sapiens | |
FG-2216 | - |
Homo sapiens | |
FG-4497 | - |
Homo sapiens | |
FG-4592 | - |
Homo sapiens | |
FKBP38 | - |
Homo sapiens | |
GSK360A | - |
Homo sapiens | |
L-mimosine | - |
Homo sapiens | |
Mn2+ | - |
Homo sapiens | |
Morg-1 | - |
Homo sapiens | |
TM6008 | - |
Homo sapiens | |
TM6089 | - |
Homo sapiens | |
Zn2+ | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
hypoxia-inducible factor-L-proline + 2-oxoglutarate + O2 | Homo sapiens | - |
hypoxia-inducible factor-trans-4-hydroxy-L-proline + succinate + CO2 | - |
? | |
additional information | Homo sapiens | isozyme PHD2 is more active on hypoxia-inducible factor-1alpha than on hypoxia-inducible factor-2alpha, whereas PHD1 and PHD3 hydroxylate hypoxia-inducible factor-2alpha more efficiently | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
mesenchymal stem cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
hypoxia-inducible factor-L-proline + 2-oxoglutarate + O2 | - |
Homo sapiens | hypoxia-inducible factor-trans-4-hydroxy-L-proline + succinate + CO2 | - |
? | |
additional information | isozyme PHD2 is more active on hypoxia-inducible factor-1alpha than on hypoxia-inducible factor-2alpha, whereas PHD1 and PHD3 hydroxylate hypoxia-inducible factor-2alpha more efficiently | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PHD | - |
Homo sapiens |
prolyl hydroxylase domain protein | - |
Homo sapiens |