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Literature summary for 1.1.1.205 extracted from

  • Jackson, R.C.; Weber, G.
    IMP dehydrogenase, an enzyme linked with proliferation and malignancy (1975), Nature, 256, 331-333.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
NAD+ 50% inhibition at 0.62 mM Rattus norvegicus
xanthosine 5'-phosphate
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
inosine 5'-phosphate + NAD+ + H2O Rattus norvegicus enzyme linked to proliferation and malignancy xanthosine 5'-phosphate + NADH
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
hepatoma
-

Source Tissue

Source Tissue Comment Organism Textmining
liver
-
Rattus norvegicus
-
spleen
-
Rattus norvegicus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
-
Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
inosine 5'-phosphate + NAD+ + H2O
-
Rattus norvegicus xanthosine 5'-phosphate + NADH
-
?
inosine 5'-phosphate + NAD+ + H2O enzyme linked to proliferation and malignancy Rattus norvegicus xanthosine 5'-phosphate + NADH
-
?

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
8.1
-
-
Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
NAD+
-
Rattus norvegicus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
additional information
-
additional information
-
Rattus norvegicus