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Ligand 1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one

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Basic Ligand Information

Molecular Structure

Picture of 1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one (click for magnification)

C₂₁H₁₆N₄OS₂

1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one

WFWGXGWFVIRPEA-UHFFFAOYSA-N

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Roles as Enzyme Ligand

Inhibitor in Enzyme-catalyzed Reactions (1 result)

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most potent inhibitor, spans the PR-ATP binding site, exhibits greater than 50% inhibition at 0.01 mM, 40% inhibition at 0.001 mM

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Enzyme Kinetic Parameters

K_i Value (1 result)

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0.002

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IC₅₀ Value (1 result)

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0.004

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References & Links

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Show Reference (1 entry)

Links to other databases for 1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one

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Release 2026.1 (March 2026)