Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Saccharomyces cerevisiae |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
17-allyl-amino-17-demethoxygeldanamycin | 0.002 mM, 20% inhibition | Saccharomyces cerevisiae | |
geldanamycin | 0.002 mM, 51% inhibition, 0.005 mM, 50% inhibition | Saccharomyces cerevisiae | |
additional information | 2 further inhibitors are found in a screen with 53440 compounds | Saccharomyces cerevisiae | |
radicicol | 0.002 mM, 88% inhibition, 0.0005 mM, 50% inhibition | Saccharomyces cerevisiae |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.51 | - |
ATP | 37°C, pH 7.4 | Saccharomyces cerevisiae |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O | Saccharomyces cerevisiae | - |
ADP + phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Saccharomyces cerevisiae | - |
- |
- |
Purification (Comment) | Organism |
---|---|
recombinant Hsp90, metal affinity, gel filtration, ion-exchange chromatography | Saccharomyces cerevisiae |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O | - |
Saccharomyces cerevisiae | ADP + phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Hsp90 | - |
Saccharomyces cerevisiae |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0078 | - |
ATP | 37°C, pH 7.4 | Saccharomyces cerevisiae |