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Literature summary for 3.5.3.15 extracted from

  • Knuckley, B.; Causey, C.P.; Pellechia, P.J.; Cook, P.F.; Thompson, P.R.
    Haloacetamidine-based inactivators of protein arginine deiminase 4 (PAD4): evidence that general acid catalysis promotes efficient inactivation (2010), ChemBioChem, 11, 161-165.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
2-chloroacetamidine
-
Homo sapiens
Cl-amidine inactivates isozyme PAD4 by the covalent modification of an active-site cysteine that is critical for catalysis Homo sapiens
F-amidine inactivates isozyme PAD4 by the covalent modification of an active-site cysteine that is critical for catalysis Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Synonyms

Synonyms Comment Organism
PAD4
-
Homo sapiens
protein arginine deiminase 4
-
Homo sapiens