Inhibitors | Comment | Organism | Structure |
---|---|---|---|
N-((1S,2R)-1-benzyl-3-cyclopropylamino-2-hydroxy-propyl)-5-(methanesulfonyl-methyl-amino)-N'-((R)-1-phenyl-ethyl)-isophthalamide | beta-secretase inhibitor IV | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | BACE1 is a transmembrane aspartyl protease with a lumenal active site | Homo sapiens | 16020 | - |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
amyloid -like PROTEIN 2 + H2O | Homo sapiens | - |
? | - |
? | |
amyloid pbeta A4 protein + H2O | Homo sapiens | - |
? | - |
? | |
amyloid-like protein 1 + H2O | Homo sapiens | - |
? | - |
? | |
basigin + H2O | Homo sapiens | - |
? | - |
? | |
beta-secretase 1 + H2O | Homo sapiens | - |
? | - |
? | |
BMP and activin membrane-bound inhibitor homolog + H2O | Homo sapiens | - |
? | - |
? | |
cache domain containing 1 + H2O | Homo sapiens | - |
? | - |
? | |
carboxypeptidase D + H2O | Homo sapiens | - |
? | - |
? | |
cation-independent mannose-6-phosphate receptor + H2O | Homo sapiens | - |
? | - |
? | |
CD166 antigen + H2O | Homo sapiens | - |
? | - |
? | |
CD276 antigen + H2O | Homo sapiens | - |
? | - |
? | |
chondroitin sulfate proteoglycan 4 + H2O | Homo sapiens | - |
? | - |
? | |
contactin-1 + H2O | Homo sapiens | - |
? | - |
? | |
cysteine-rich motor neuron 1 protein + H2O | Homo sapiens | - |
? | - |
? | |
desmoglein 2 + H2O | Homo sapiens | - |
? | - |
? | |
disintegrin and metalloproteinase domain-containing protein 10 + H2O | Homo sapiens | - |
? | - |
? | |
ephrin type-A receptor 2 + H2O | Homo sapiens | - |
? | - |
? | |
ephrin type-A receptor 4 + H2O | Homo sapiens | - |
? | - |
? | |
ephrin type-A receptor 7 + H2O | Homo sapiens | - |
? | - |
? | |
ephrin-A5 + H2O | Homo sapiens | - |
? | - |
? | |
glypican-3 + H2O | Homo sapiens | - |
? | - |
? | |
Golgi apparatus protein 1 + H2O | Homo sapiens | - |
? | - |
? | |
Golgi phosphoprotein 4 + H2O | Homo sapiens | - |
? | - |
? | |
hepatocyte growth factor receptor + H2O | Homo sapiens | - |
? | - |
? | |
HLA class I histocompatibility antigen (combined) + H2O | Homo sapiens | - |
? | - |
? | |
interleukin-6 receptor beta chain + H2O | Homo sapiens | - |
? | - |
? | |
Jagged-1 + H2O | Homo sapiens | - |
? | - |
? | |
Kunitz-type protease inhibitor 2 + H2O | Homo sapiens | - |
? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 1 + H2O | Homo sapiens | - |
? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 2 + H2O | Homo sapiens | - |
? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 3 + H2O | Homo sapiens | - |
? | - |
? | |
leucine-rich repeat-containing protein 33 + H2O | Homo sapiens | - |
? | - |
? | |
low-density lipoprotein receptor-related protein 11 + H2O | Homo sapiens | - |
? | - |
? | |
low-density lipoprotein receptor-related protein 4 + H2O | Homo sapiens | - |
? | - |
? | |
neogenin + H2O | Homo sapiens | - |
? | - |
? | |
netrin receptor UNC5C + H2O | Homo sapiens | - |
? | - |
? | |
neuronal cell adhesion molecule 1 + H2O | Homo sapiens | - |
? | - |
? | |
neuronal cell adhesion molecule L1 + H2O | Homo sapiens | - |
? | - |
? | |
peptidyl-glycine alpha-amidating monooxygenase + H2O | Homo sapiens | - |
? | - |
? | |
plexin domain-containing protein 2 + H2O | Homo sapiens | - |
? | - |
? | |
podocalyxin-like protein 1 + H2O | Homo sapiens | - |
? | - |
? | |
poliovirus receptor type I + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin 21 + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin 7 + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin gamma A11 + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin gamma A5 + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin gamma A8 + H2O | Homo sapiens | - |
? | - |
? | |
protocadherin gamma C3 + H2O | Homo sapiens | - |
? | - |
? | |
protogenin + H2O | Homo sapiens | - |
? | - |
? | |
receptor protein tyrosine kinase variant EPHB4V1 + H2O | Homo sapiens | - |
? | - |
? | |
receptor-type tyrosin-protein phosphatase S + H2O | Homo sapiens | - |
? | - |
? | |
roundabout homolog 1 + H2O | Homo sapiens | - |
? | - |
? | |
roundabout homolog 2 + H2O | Homo sapiens | - |
? | - |
? | |
seizure 6-like protein 2 + H2O | Homo sapiens | - |
? | - |
? | |
semaphorin-4B + H2O | Homo sapiens | - |
? | - |
? | |
semaphorin-4C + H2O | Homo sapiens | - |
? | - |
? | |
semaphorin-6A + H2O | Homo sapiens | - |
? | - |
? | |
semaphorin-6D + H2O | Homo sapiens | - |
? | - |
? | |
sidekick-1 + H2O | Homo sapiens | - |
? | - |
? | |
sidekick-2 + H2O | Homo sapiens | - |
? | - |
? | |
sortilin type I + H2O | Homo sapiens | - |
? | - |
? | |
sortilin-related receptor type I + H2O | Homo sapiens | - |
? | - |
? | |
syndecan-4 + H2O | Homo sapiens | - |
? | - |
? | |
T-cell immunomodulatory protein + H2O | Homo sapiens | - |
? | - |
? | |
toll-like receptor 9 + H2O | Homo sapiens | - |
? | - |
? | |
trans-Golgi network integral membrane protein 2 + H2O | Homo sapiens | - |
? | - |
? | |
transmembrane protein 132A + H2O | Homo sapiens | - |
? | - |
? | |
tumor necrosis factor receptor superfamily member 21 + H2O | Homo sapiens | - |
? | - |
? | |
vesicular integral-membrane protein VIP36 + H2O | Homo sapiens | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Posttranslational Modification | Comment | Organism |
---|---|---|
glycoprotein | - |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HEK-293FT cell | - |
Homo sapiens | - |
HeLa cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
amyloid -like PROTEIN 2 + H2O | - |
Homo sapiens | ? | - |
? | |
amyloid pbeta A4 protein + H2O | - |
Homo sapiens | ? | - |
? | |
amyloid-like protein 1 + H2O | - |
Homo sapiens | ? | - |
? | |
basigin + H2O | - |
Homo sapiens | ? | - |
? | |
beta-secretase 1 + H2O | - |
Homo sapiens | ? | - |
? | |
BMP and activin membrane-bound inhibitor homolog + H2O | - |
Homo sapiens | ? | - |
? | |
cache domain containing 1 + H2O | - |
Homo sapiens | ? | - |
? | |
carboxypeptidase D + H2O | - |
Homo sapiens | ? | - |
? | |
cation-independent mannose-6-phosphate receptor + H2O | - |
Homo sapiens | ? | - |
? | |
CD166 antigen + H2O | - |
Homo sapiens | ? | - |
? | |
CD276 antigen + H2O | - |
Homo sapiens | ? | - |
? | |
chondroitin sulfate proteoglycan 4 + H2O | - |
Homo sapiens | ? | - |
? | |
contactin-1 + H2O | - |
Homo sapiens | ? | - |
? | |
cysteine-rich motor neuron 1 protein + H2O | - |
Homo sapiens | ? | - |
? | |
desmoglein 2 + H2O | - |
Homo sapiens | ? | - |
? | |
disintegrin and metalloproteinase domain-containing protein 10 + H2O | - |
Homo sapiens | ? | - |
? | |
ephrin type-A receptor 2 + H2O | - |
Homo sapiens | ? | - |
? | |
ephrin type-A receptor 4 + H2O | - |
Homo sapiens | ? | - |
? | |
ephrin type-A receptor 7 + H2O | - |
Homo sapiens | ? | - |
? | |
ephrin-A5 + H2O | - |
Homo sapiens | ? | - |
? | |
glypican-3 + H2O | - |
Homo sapiens | ? | - |
? | |
Golgi apparatus protein 1 + H2O | - |
Homo sapiens | ? | - |
? | |
Golgi phosphoprotein 4 + H2O | - |
Homo sapiens | ? | - |
? | |
hepatocyte growth factor receptor + H2O | - |
Homo sapiens | ? | - |
? | |
HLA class I histocompatibility antigen (combined) + H2O | - |
Homo sapiens | ? | - |
? | |
interleukin-6 receptor beta chain + H2O | - |
Homo sapiens | ? | - |
? | |
Jagged-1 + H2O | - |
Homo sapiens | ? | - |
? | |
Kunitz-type protease inhibitor 2 + H2O | - |
Homo sapiens | ? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 1 + H2O | - |
Homo sapiens | ? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 2 + H2O | - |
Homo sapiens | ? | - |
? | |
leucin-rich repeats and immunoglobulin-like domains protein 3 + H2O | - |
Homo sapiens | ? | - |
? | |
leucine-rich repeat-containing protein 33 + H2O | - |
Homo sapiens | ? | - |
? | |
low-density lipoprotein receptor-related protein 11 + H2O | - |
Homo sapiens | ? | - |
? | |
low-density lipoprotein receptor-related protein 4 + H2O | - |
Homo sapiens | ? | - |
? | |
neogenin + H2O | - |
Homo sapiens | ? | - |
? | |
netrin receptor UNC5C + H2O | - |
Homo sapiens | ? | - |
? | |
neuronal cell adhesion molecule 1 + H2O | - |
Homo sapiens | ? | - |
? | |
neuronal cell adhesion molecule L1 + H2O | - |
Homo sapiens | ? | - |
? | |
peptidyl-glycine alpha-amidating monooxygenase + H2O | - |
Homo sapiens | ? | - |
? | |
plexin domain-containing protein 2 + H2O | - |
Homo sapiens | ? | - |
? | |
podocalyxin-like protein 1 + H2O | - |
Homo sapiens | ? | - |
? | |
poliovirus receptor type I + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin 21 + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin 7 + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin gamma A11 + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin gamma A5 + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin gamma A8 + H2O | - |
Homo sapiens | ? | - |
? | |
protocadherin gamma C3 + H2O | - |
Homo sapiens | ? | - |
? | |
protogenin + H2O | - |
Homo sapiens | ? | - |
? | |
receptor protein tyrosine kinase variant EPHB4V1 + H2O | - |
Homo sapiens | ? | - |
? | |
receptor-type tyrosin-protein phosphatase S + H2O | - |
Homo sapiens | ? | - |
? | |
roundabout homolog 1 + H2O | - |
Homo sapiens | ? | - |
? | |
roundabout homolog 2 + H2O | - |
Homo sapiens | ? | - |
? | |
seizure 6-like protein 2 + H2O | - |
Homo sapiens | ? | - |
? | |
semaphorin-4B + H2O | - |
Homo sapiens | ? | - |
? | |
semaphorin-4C + H2O | - |
Homo sapiens | ? | - |
? | |
semaphorin-6A + H2O | - |
Homo sapiens | ? | - |
? | |
semaphorin-6D + H2O | - |
Homo sapiens | ? | - |
? | |
sidekick-1 + H2O | - |
Homo sapiens | ? | - |
? | |
sidekick-2 + H2O | - |
Homo sapiens | ? | - |
? | |
sortilin type I + H2O | - |
Homo sapiens | ? | - |
? | |
sortilin-related receptor type I + H2O | - |
Homo sapiens | ? | - |
? | |
syndecan-4 + H2O | - |
Homo sapiens | ? | - |
? | |
T-cell immunomodulatory protein + H2O | - |
Homo sapiens | ? | - |
? | |
toll-like receptor 9 + H2O | - |
Homo sapiens | ? | - |
? | |
trans-Golgi network integral membrane protein 2 + H2O | - |
Homo sapiens | ? | - |
? | |
transmembrane protein 132A + H2O | - |
Homo sapiens | ? | - |
? | |
tumor necrosis factor receptor superfamily member 21 + H2O | - |
Homo sapiens | ? | - |
? | |
vesicular integral-membrane protein VIP36 + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
BACE1 | - |
Homo sapiens |
beta-secretase | - |
Homo sapiens |