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Literature summary for 3.4.23.16 extracted from

  • Bihani, S.C.; Das, A.; Prashar, V.; Ferrer, J.L.; Hosur, M.V.
    Resistance mechanism revealed by crystal structures of unliganded nelfinavir-resistant HIV-1 protease non-active site mutants N88D and N88S (2009), Biochem. Biophys. Res. Commun., 389, 295-300.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
-
Human immunodeficiency virus 1

Crystallization (Commentary)

Crystallization (Comment) Organism
hanging-drop vapor diffusion method Human immunodeficiency virus 1

Protein Variants

Protein Variants Comment Organism
N88D non-active site region, nelfinavir resistent Human immunodeficiency virus 1
N88S non-active site region, nelfinavir resistent Human immunodeficiency virus 1

Inhibitors

Inhibitors Comment Organism Structure
nelfinavir
-
Human immunodeficiency virus 1

Organism

Organism UniProt Comment Textmining
Human immunodeficiency virus 1
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Human immunodeficiency virus 1

Subunits

Subunits Comment Organism
homodimer crystal structure analysis Human immunodeficiency virus 1

Synonyms

Synonyms Comment Organism
HIV-1 protease
-
Human immunodeficiency virus 1