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Literature summary for 3.4.23.15 extracted from

  • Whaley-Connell, A.; Nistala, R.; Habibi, J.; Hayden, M.R.; Schneider, R.I.; Johnson, M.S.; Tilmon, R.; Rehmer, N.; Ferrario, C.M.; Sowers, J.R.
    Comparative effect of direct renin inhibition and AT1R blockade on glomerular filtration barrier injury in the transgenic Ren2 rat (2010), Am. J. Physiol. Renal Physiol., 298, F655-F661.
    View publication on PubMedView publication on EuropePMC

Application

Application Comment Organism
medicine blockade of renin activation is a therapeutic target to prevent glomerular injury and associated proteinuria Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
aliskiren potent direct renin inhibitor Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
angiotensinogen + H2O Rattus norvegicus
-
angiotensin I + angiotensinogen propeptide
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
angiotensinogen + H2O
-
Rattus norvegicus angiotensin I + angiotensinogen propeptide
-
?

General Information

General Information Comment Organism
metabolism renin is the rate-limiting step in angiotensin II generation Rattus norvegicus